4-Benzyl- and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones, a New Family of Potent Anti-HIV Agents: Optimization and in Vitro Evaluation against Clinically Important HIV Mutant Strains-Reference-Cited by-同舟云学术

4-Benzyl- and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones, a New Family of Potent Anti-HIV Agents: Optimization and in Vitro Evaluation against Clinically Important HIV Mutant Strains

Published:2004-09-29 Issue:22 Volume:47 Page:5501-5514
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Benjahad Abdellah¹,Courté Karine¹,Guillemont Jérôme¹,Mabire Dominique¹,Coupa Sophie¹,Poncelet Alain¹,Csoka Imre¹,Andries Koen¹,Pauwels Rudi¹,de Béthune Marie-Pierre¹,Monneret Claude¹,Bisagni Emile¹,Nguyen Chi Hung¹,Grierson David S.¹

Affiliation:

1. UMR 176 CNRS-Institut Curie, Laboratoire de Pharmacochimie, Section de Recherche, Batiment 110, Centre Universitaire, 91405 Orsay, France, Johnson&Johnson Pharmaceutical Research and Development, Medicinal Chemistry Department, Campus de Maigremont BP315, Val de Reuil, France, Johnson&Johnson Pharmaceutical Research and Development, Virology Drug Discovery, Tumhoutseweg 30 B-2340 Beerse, Belgium, and TIBOTEC, Generaal De Wittelaan L 11 B3, B-2800 Mechelen, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0407658

Reference54 articles.

1. Decline in the AIDS and death rates in the EuroSIDA study: an observational study

2. HIV chemotherapy

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4. Novel compounds in preclinical/early clinical development for the treatment of HIV infections

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