Structural Analysis of ARC-Type Inhibitor (ARC-1034) Binding to Protein Kinase A Catalytic Subunit and Rational Design of Bisubstrate Analogue Inhibitors of Basophilic Protein Kinases-Reference-Cited by-同舟云学术

Structural Analysis of ARC-Type Inhibitor (ARC-1034) Binding to Protein Kinase A Catalytic Subunit and Rational Design of Bisubstrate Analogue Inhibitors of Basophilic Protein Kinases

Published:2008-12-29 Issue:2 Volume:52 Page:308-321
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lavogina Darja¹,Lust Marje¹,Viil Indrek¹,König Norbert¹,Raidaru Gerda¹,Rogozina Jevgenia¹,Enkvist Erki¹,Uri Asko¹,Bossemeyer Dirk¹

Affiliation:

1. Institute of Chemistry, 2 Jakobi Street, 51014 Tartu, Estonia, Group of Structural Biochemistry, German Cancer Research Centre, Im Neuenheimer Feld 280, 69120 Heidelberg, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800797n

Reference54 articles.

1. The Protein Kinase Complement of the Human Genome

2. REVIEW Structural Insights Into AGC Kinase Inhibition

3. Protein kinases — the major drug targets of the twenty-first century?

4. Protein Kinase Inhibitors: Insights into Drug Design from Structure

5. Tracking Cell Signaling Protein Expression and Phosphorylation by Innovative Proteomic Solutions

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