Synthesis and Structure–Activity Relationship Studies of Conformationally Flexible Tetrahydroisoquinolinyl Triazole Carboxamide and Triazole Substituted Benzamide Analogues as σ2 Receptor Ligands-Reference-Cited by-同舟云学术

Synthesis and Structure–Activity Relationship Studies of Conformationally Flexible Tetrahydroisoquinolinyl Triazole Carboxamide and Triazole Substituted Benzamide Analogues as σ2 Receptor Ligands

Published:2014-05-12 Issue:10 Volume:57 Page:4239-4251
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bai Suping¹²,Li Shihong¹,Xu Jinbin¹,Peng Xin¹,Sai Kiran¹,Chu Wenhua¹,Tu Zhude¹,Zeng Chenbo¹,Mach Robert H.¹

Affiliation:

1. Department of Radiology, Washington University School of Medicine, St. Louis, Missouri 63110, United States

2. School of Pharmacy, Xinxiang Medical University, Xinxiang, Henan 453003, China

Funder

U.S. Department of Energy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5001453

Reference68 articles.

1. Autoradiographic distribution of [3H](+)-pentazocine and [3H]1,3-di-o-tolylguanidine (DTG) binding sites in guinea pig brain: a comparative study

2. Rat liver and kidney contain high densities of σ1 and σ2 receptors: characterization by ligand binding and photoaffinity labeling

3. A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain

4. A proposal for the classification of sigma binding sites

Cited by 36 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis, spectroscopic, electrochemistry and antioxidant properties of benzofuroxan and 2H-benzimidazole 1,3-dioxide derivatives: Effects of conjugation with electron-acceptor 1,2,3-triazolyl-1,2,4-oxadiazole;Journal of Molecular Structure;2024-09

2. Shedding Light on the D₁‐Like Receptors: A Fluorescence‐Based Toolbox for Visualization of the D₁ and D₅ Receptors**;ChemBioChem;2023-11-20

3. Shedding Light on the D₁-Like Receptors: A Fluorescence-Based Toolbox for Visualization of the D₁and D₅Receptors;2023-09-25

4. Continuous Flow Synthesis of N-Sulfonyl-1,2,3-triazoles for Tandem Relay Cu/Rh Dual Catalysis;The Journal of Organic Chemistry;2023-01-04

5. Magnetic carbon–based nanocomposite decorated with palladium complex for co-delivery of DOX/pCRISPR;Journal of Drug Delivery Science and Technology;2022-12