Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain-Reference-Cited by-同舟云学术

Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain

Published:2015-02-11 Issue:4 Volume:58 Page:1915-1928
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cuzzucoli Crucitti Giuliana¹,Métifiot Mathieu²,Pescatori Luca¹,Messore Antonella¹,Madia Valentina Noemi¹,Pupo Giovanni¹,Saccoliti Francesco¹,Scipione Luigi¹,Tortorella Silvano¹,Esposito Francesca³,Corona Angela³,Cadeddu Marta³,Marchand Christophe²,Pommier Yves²,Tramontano Enzo³,Costi Roberta¹,Di Santo Roberto¹

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, “Sapienza” Università di Roma, Rome, I-00185, Italy

2. Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Building 37, Room 5068, Bethesda, Maryland 20892-4255, United States

3. Department of Life and Environmental Sciences, University of Cagliari, Cagliari, 09124, Italy

Funder

National Cancer Institute

European Commission

Ministero dell'Istruzione, dell'Università e della Ricerca

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501799k

Reference48 articles.