Structural Insights into the Molecular Mechanism of Vitamin D Receptor Activation by Lithocholic Acid Involving a New Mode of Ligand Recognition-Reference-Cited by-同舟云学术

Structural Insights into the Molecular Mechanism of Vitamin D Receptor Activation by Lithocholic Acid Involving a New Mode of Ligand Recognition

Published:2014-05-21 Issue:11 Volume:57 Page:4710-4719
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Belorusova Anna Y.¹,Eberhardt Jérôme¹,Potier Noëlle²,Stote Roland H.¹,Dejaegere Annick¹,Rochel Natacha¹

Affiliation:

1. Department of Integrative Structural Biology, Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Institut National de Santé et de Recherche Médicale (INSERM) U964, Centre National de Recherche Scientifique (CNRS) UMR 7104, Université de Strasbourg, 67404 Illkirch, France

2. Institut de Chimie LC3, CNRS, UMR 7177, 67008 Strasbourg, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5002524

Reference49 articles.

1. Vitamin D receptor (VDR)-mediated actions of 1α,25(OH)2vitamin D3: Genomic and non-genomic mechanisms

2. The vitamin D receptor as a therapeutic target

3. Vitamin D Receptor As an Intestinal Bile Acid Sensor

4. Structural Determinants for Vitamin D Receptor Response to Endocrine and Xenobiotic Signals

5. Selective activation of vitamin D receptor by lithocholic acid acetate, a bile acid derivative

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