Design of Non-nucleoside Inhibitors of HIV-1 Reverse Transcriptase with Improved Drug Resistance Properties. 2.-Reference-Cited by-同舟云学术

Design of Non-nucleoside Inhibitors of HIV-1 Reverse Transcriptase with Improved Drug Resistance Properties. 2.

Published:2004-10-23 Issue:24 Volume:47 Page:5923-5936
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Freeman George A.¹,Andrews C. Webster¹,Hopkins Andrew L.¹,Lowell Gina S.¹,Schaller Lee T.¹,Cowan Jill R.¹,Gonzales Stephen S.¹,Koszalka George W.¹,Hazen Richard J.¹,Boone Lawrence R.¹,Ferris Rob G.¹,Creech Katrina L.¹,Roberts Grace B.¹,Short Steven A.¹,Weaver Kurt¹,Reynolds David J.¹,Milton John¹,Ren Jingshan¹,Stuart David I.¹,Stammers David K.¹,Chan Joseph H.¹

Affiliation:

1. GlaxoSmithKline Research and Development, 5 Moore Drive, Research Triangle Park, North Carolina 27709, Division of Structural Biology, The Wellcome Trust Centre for Human Genetics, University of Oxford, Roosevelt Drive, Oxford, OX3 7BN, UK, and Oxford Centre for Molecular Sciences, New Chemistry Building, University of Oxford, South Parks Road, Oxford, OX1 3QT, UK

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm040072r

Reference32 articles.

1. Viral RNA-dependent DNA Polymerase: RNA-dependent DNA Polymerase in Virions of RNA Tumour Viruses

2. Inhibition of HIV-1 Replication by a Nonnucleoside Reverse Transcriptase Inhibitor

3. L-743, 726 (DMP-266): a novel, highly potent nonnucleoside inhibitor of the human immunodeficiency virus type 1 reverse transcriptase

4. Unique features in the structure of the complex between HIV-1 reverse transcriptase and the bis(heteroaryl)piperazine (BHAP) U-90152 explain resistance mutations for this nonnucleoside inhibitor

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