β-Lactams Derived from a Carbapenem Chiron Are Selective Inhibitors of Human Fatty Acid Amide Hydrolase versus Human Monoacylglycerol Lipase-Reference-Cited by-同舟云学术

β-Lactams Derived from a Carbapenem Chiron Are Selective Inhibitors of Human Fatty Acid Amide Hydrolase versus Human Monoacylglycerol Lipase

Published:2009-10-30 Issue:22 Volume:52 Page:7054-7068
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Feledziak Marion¹²,Michaux Catherine³,Urbach Allan¹,Labar Geoffray²,Muccioli Giulio G.²,Lambert Didier M.²,Marchand-Brynaert Jacqueline¹

Affiliation:

1. Unité de Chimie Organique et Médicinale, Université Catholique de Louvain, Bâtiment Lavoisier, Place Louis Pasteur 1, B-1348 Louvain-La-Neuve, Belgium

2. Unité de Chimie Pharmaceutique et de Radiopharmacie, Louvain Drug Research Institute, Université Catholique de Louvain, Avenue E. Mounier 73.40, B-1200 Bruxelles, Belgium

3. Laboratoire de Chimie Biologique Structurale, Facultés Universitaires Notre-Dame de la Paix, rue de Bruxelles 61, B-5000 Namur, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9008532

Reference58 articles.

1. Synthesis and evaluation of N1/C4-substituted β-lactams as PPE and HLE inhibitors

2. Design, Synthesis, and Proposed Active Site Binding Analysis of Monocyclic 2-Azetidinone Inhibitors of Prostate Specific Antigen

3. Azetidin-2-one derivatives as inhibitors of thrombin

4. Design and synthesis of monocyclic β-lactams as mechanism-based inhibitors of human cytomegalovirus protease

5. Penicillins

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