A New Quantitative Cell-Based Assay Reveals Unexpected Microtubule Stabilizing Activity of Certain Kinase Inhibitors, Clinically Approved or in the Process of Approval-Reference-Cited by-同舟云学术

A New Quantitative Cell-Based Assay Reveals Unexpected Microtubule Stabilizing Activity of Certain Kinase Inhibitors, Clinically Approved or in the Process of Approval

Published:2020-04-30 Issue: Volume:11 Page:
ISSN:1663-9812
Container-title:Frontiers in Pharmacology
language:
Short-container-title:Front. Pharmacol.

Author:

Ramirez-Rios Sacnicte,Michallet Sophie,Peris Leticia,Barette Caroline,Rabat Clotilde,Feng Yangbo,Fauvarque Marie-Odile,Andrieux Annie,Sadoul Karin,Lafanechère Laurence

Funder

Institut National Du Cancer

Publisher

Frontiers Media SA

Subject

Pharmacology (medical),Pharmacology

Reference63 articles.

1. Mps1 is a kinetochore-associated kinase essential for the vertebrate mitotic checkpoint;Abrieu;Cell,2001

2. Vasohibins/SVBP are tubulin carboxypeptidases (TCP) that regulate neuron differentiation;Aillaud;Science,2017

3. Tivantinib (ARQ 197) Exhibits Antitumor Activity by Directly Interacting with Tubulin and Overcomes ABC Transporter–Mediated Drug Resistance;Aoyama;Mol. Cancer Ther.,2014

4. Deconvolution of Buparlisib’s mechanism of action defines specific PI3K and tubulin inhibitors for therapeutic intervention;Bohnacker;Nat. Commun.,2017

5. Masitinib (AB1010), a Potent and Selective Tyrosine Kinase Inhibitor Targeting KIT;Dubreuil;PloS One,2009

Cited by 10 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Mechanisms of cytotoxic activity of pyrrole-carboxamides against multidrug-resistant tumor cell sublines;Advances in Molecular Oncology;2023-10-09

2. Quantitative analysis of the effect of microtubule-targeting drugs on the microtubule cytoskeleton of breast cancer cells with different invasive properties;Comptes Rendus. Chimie;2023-09-19

3. Design, synthesis and biological evaluation of quinoline-2-carbonitrile-based hydroxamic acids as dual tubulin polymerization and histone deacetylases inhibitors;European Journal of Medicinal Chemistry;2022-10

4. The microtubule cytoskeleton: An old validated target for novel therapeutic drugs;Frontiers in Pharmacology;2022-09-15

5. Morphological profiling by means of the Cell Painting assay enables identification of tubulin-targeting compounds;Cell Chemical Biology;2021-12