NUC041, a Prodrug of the DNA Methytransferase Inhibitor 5-aza-2′,2′-Difluorodeoxycytidine (NUC013), Leads to Tumor Regression in a Model of Non-Small Cell Lung Cancer
Author:
Publisher
MDPI AG
Subject
Drug Discovery,Pharmaceutical Science,Molecular Medicine
Link
http://www.mdpi.com/1424-8247/11/2/36/pdf
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2. 5-Aza-4′-thio-2′-deoxycytidine, a New Orally Bioavailable Nontoxic “Best-in-Class”: DNA Methyltransferase 1–Depleting Agent in Clinical Development;Journal of Pharmacology and Experimental Therapeutics;2021-09-09
3. Regioselective synthesis and anticancer evaluation of H2O2-activable nucleosides;Chemical Communications;2020
4. Pharmacoepigenetics of Novel Nucleoside DNA Methyltransferase Inhibitors;Pharmacoepigenetics;2019
5. Pharmacoepigenetic Processors: Epigenetic Drugs, Drug Resistance, Toxicoepigenetics, and Nutriepigenetics;Pharmacoepigenetics;2019
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