Non-Imidazole Histamine H3 Ligands. Part VII. Synthesis, In Vitro and In Vivo Characterization of 5-Substituted-2-thiazol-4-n-propylpiperazines-Reference-Cited by-同舟云学术

Non-Imidazole Histamine H3 Ligands. Part VII. Synthesis, In Vitro and In Vivo Characterization of 5-Substituted-2-thiazol-4-n-propylpiperazines

Published:2018-02-03 Issue:2 Volume:23 Page:326
ISSN:1420-3049
Container-title:Molecules
language:en
Short-container-title:Molecules

Author:

Guryn Roman,Staszewski Marek,Stasiak Anna,McNaught Flores Daniel,Fogel Wiesława,Leurs Rob,Walczyński Krzysztof

Publisher

MDPI AG

Subject

Chemistry (miscellaneous),Analytical Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Molecular Medicine,Drug Discovery,Pharmaceutical Science

Link

http://www.mdpi.com/1420-3049/23/2/326/pdf

Reference46 articles.

1. The physiology of brain histamine

2. Three histamine receptors (H1, H2 and H3) visualized in the brain of human and non-human primates

3. A detailed autoradiographic mapping of histamine H3 receptors in rat brain areas

4. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

5. Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

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