4-Hydroxypiperidines and Their Flexible 3-(Amino)propyloxy Analogues as Non-Imidazole Histamine H3 Receptor Antagonist: Further Structure–Activity Relationship Exploration and In Vitro and In Vivo Pharmacological Evaluation-Reference-Cited by-同舟云学术

4-Hydroxypiperidines and Their Flexible 3-(Amino)propyloxy Analogues as Non-Imidazole Histamine H3 Receptor Antagonist: Further Structure–Activity Relationship Exploration and In Vitro and In Vivo Pharmacological Evaluation

Published:2018-04-19 Issue:4 Volume:19 Page:1243
ISSN:1422-0067
Container-title:International Journal of Molecular Sciences
language:en
Short-container-title:IJMS

Author:

Olszewska Beata,Stasiak Anna,McNaught Flores Daniel,Fogel Wiesława,Leurs Rob,Walczyński Krzysztof

Publisher

MDPI AG

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Computer Science Applications,Spectroscopy,Molecular Biology,General Medicine,Catalysis

Link

http://www.mdpi.com/1422-0067/19/4/1243/pdf

Reference47 articles.

1. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

2. H3-Receptors Control Histamine Release in Human Brain

3. Cloning and Functional Expression of the Human Histamine H3Receptor

4. Presynaptic H3Autoreceptors Modulate Histamine Synthesis through cAMP Pathway

5. Histamine H3receptors mediate inhibition of noradrenaline release from intestinal sympathetic nerves

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