Structural Hypervariability of the Two Human Protein Kinase CK2 Catalytic Subunit Paralogs Revealed by Complex Structures with a Flavonol- and a Thieno[2,3-d]pyrimidine-Based Inhibitor
Author:
Funder
Deutsche Forschungsgemeinschaft
National Academy of Sciences of Ukraine
Publisher
MDPI AG
Subject
Drug Discovery,Pharmaceutical Science,Molecular Medicine
Link
http://www.mdpi.com/1424-8247/10/1/9/pdf
Reference49 articles.
1. The Conformational Plasticity of Protein Kinases
2. Crystal structures of the kinase domain of c-Abl in complex with the small molecule inhibitors PD173955 and imatinib (STI-571);Nagar;Cancer Res.,2002
3. Inhibition of p38 MAP kinase by utilizing a novel allosteric binding site
4. Mutagenesis of p38α MAP Kinase Establishes Key Roles of Phe169 in Function and Structural Dynamics and Reveals a Novel DFG-OUT State
5. A conserved protonation-dependent switch controls drug binding in the Abl kinase
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