The A3adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches-Reference-Cited by-同舟云学术

The A3adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches

Published:2011-11-16 Issue:2 Volume:33 Page:235-335
ISSN:0198-6325
Container-title:Medicinal Research Reviews
language:en
Short-container-title:Med. Res. Rev.

Author:

Cheong Siew Lee¹,Federico Stephanie²,Venkatesan Gopalakrishnan¹,Mandel Alexander Laurence¹,Shao Yi-Ming¹³,Moro Stefano⁴,Spalluto Giampiero²,Pastorin Giorgia¹³

Affiliation:

1. Department of Pharmacy; National University of Singapore; 3 Science Drive 2 Singapore 117543 Singapore

2. Dipartimento di Scienze Farmaceutiche; Università degli Studi di Trieste; Piazzale Europa 1 I-34127 Trieste Italy

3. NUS Graduate School for Integrative Sciences and Engineering; Centre for Life Sciences (CeLS); 28 Medical Drive ♯05-01 Singapore 117456 Singapore

4. Molecular Modeling Section (MMS); Dipartimento di Scienze Farmaceutiche; Università di Padova; via Marzolo 5 I-35131 Padova Italy

Publisher

Wiley

Subject

Drug Discovery,Pharmacology,Molecular Medicine

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/med.20254/fullpdf

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3. Modeling the adenosine receptors: Comparison of binding domains of A2A agonist and antagonist;Kim;J Med Chem,2003

4. Identification of threonine residues controlling the agonist-dependent phosphorylation and desensitization of the rat adenosine receptor;Palmer;Mol Pharmacol,2000

5. A3 adenosine receptors in human astrocytoma cells: Agonist-mediated desensitization, internalization, and down-regulation;Trincavelli;Mol Pharmacol,2002

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