New cancer drugs targeting the biosynthesis of estrogens and androgens
Author:
Publisher
Wiley
Subject
Drug Discovery
Reference129 articles.
1. Steroidal and non-steroidal inhibitors of steroid 5α-reductase;Abell;Curr Med Chem,1995
2. Control of secretion and function of C19-delta 5-steroids of the human adrenal gland;Adams;Mol Cell Endocrinol,1985
3. Review of estrone sulfatase and its inhibitors-an important new target against hormone dependent breast cancer;Ahmed;Curr Med Chem,2002
4. The estradiol pharmacophore: ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site;Anstead;Steroids,1997
5. Inhibitors of steroidal cytochrome p450 enzymes as targets for drug development;Baston;Recent Patents Anticancer Drug Discov,2007
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