Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels-Reference-Cited by-同舟云学术

Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels

Published:2021-10-05 Issue:23 Volume:16 Page:3588-3599
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Milani Gualtiero¹,Cavalluzzi Maria Maddalena¹^ORCID,Altamura Concetta²,Santoro Antonella³,Perrone Mariagrazia¹,Muraglia Marilena¹,Colabufo Nicola Antonio¹,Corbo Filomena¹,Casalino Elisabetta⁴,Franchini Carlo¹,Pisano Isabella³,Desaphy Jean‐François²,Carrieri Antonio¹,Carocci Alessia¹,Lentini Giovanni¹

Affiliation:

1. Department of Pharmacy – Pharmaceutical Sciences University of Bari Aldo Moro Via E. Orabona 4 70125 Bari Italy

2. Department of Biomedical Sciences and Human Oncology School of Medicine University of Bari Aldo Moro Policlinico Piazza Giulio Cesare 70124 Bari Italy

3. Department of Bioscience, Biotechnology and Biopharmaceutics University of Bari Aldo Moro Via Orabona 4 70125 Bari Italy

4. Department of Veterinary Medicine University of Bari Aldo Moro Via E. Orabona 4 70125 Bari Italy

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202100496

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