Development of Riluzole Analogs with Improved Use-Dependent Inhibition of Skeletal Muscle Sodium Channels-Reference-Cited by-同舟云学术

Development of Riluzole Analogs with Improved Use-Dependent Inhibition of Skeletal Muscle Sodium Channels

Published:2023-06-23 Issue:7 Volume:14 Page:999-1008
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Farinato Alessandro¹^ORCID,Cavalluzzi Maria Maddalena²^ORCID,Altamura Concetta³,Campanale Carmen³,Laghetti Paola³,Saltarella Ilaria³,Delre Pietro⁴,Barbault Arthur⁴,Tarantino Nancy¹,Milani Gualtiero²,Rotondo Natalie Paola²,Di Cesare Mannelli Lorenzo⁵,Ghelardini Carla⁵,Pierno Sabata¹,Mangiatordi Giuseppe Felice⁴^ORCID,Lentini Giovanni²,Desaphy Jean-François³

Affiliation:

1. Section of Pharmacology, Department of Pharmacy − Drug Sciences, University of Bari Aldo Moro, 70125 Bari, Italy

2. Section of Medicinal Chemistry, Department of Pharmacy − Drug Sciences, University of Bari Aldo Moro, 70125 Bari, Italy

3. Section of Pharmacology, Department of Precision and Regenerative Medicine, School of Medicine, University of Bari Aldo Moro, 70124 Bari, Italy

4. CNR − Institute of Crystallography, via Amendola 122/o, 70126 Bari, Italy

5. Department NEUROFARBA - Pharmaceutical and Nutraceutical Section, University of Firenze, 50139 Florence, Italy

Funder

French Muscular Dystrophy Association

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.3c00224

Reference31 articles.

1. A Controlled Trial of Riluzole in Amyotrophic Lateral Sclerosis

2. Dose-ranging study of riluzole in amyotrophic lateral sclerosis

3. Effects of Benzothiazolamines on Voltage-Gated Sodium Channels

4. From Riluzole to Dexpramipexole via Substituted-Benzothiazole Derivatives for Amyotrophic Lateral Sclerosis Disease Treatment: Case Studies

5. Substituted 2-Benzothiazolamines as Sodium Flux Inhibitors: Quantitative Structure-Activity Relationships and Anticonvulsant Activity

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