Synthesis of Aminoethyl‐Substituted Piperidine Derivatives as σ <sub>1</sub> Receptor Ligands with Antiproliferative Properties-Reference-Cited by-同舟云学术

Synthesis of Aminoethyl‐Substituted Piperidine Derivatives as σ ₁ Receptor Ligands with Antiproliferative Properties

Published:2022-02-09 Issue:7 Volume:17 Page:
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Holtschulte Catharina¹,Börgel Frederik¹,Westphälinger Stefanie¹,Schepmann Dirk¹,Civenni Gianluca²,Laurini Erik³,Marson Domenico³,Catapano Carlo V.²,Pricl Sabrina³⁴,Wünsch Bernhard¹⁵^ORCID

Affiliation:

1. Institut für Pharmazeutische und Medizinische Chemie Westfälische Wilhelms-Universität Münster Corrensstraße 48 48149 Münster Germany

2. Institute of Oncology Research Università della Svizzera Italiana (USI) Via Vincenzo Vela 6 6500 Bellinzona Switzerland

3. Molecular Biology and Nanotechnology Laboratory (MolBNL@UniTS), DEA University of Trieste 34127 Trieste Italy

4. Department of General Biophysics Faculty of Biology and Environmental Protection University of Lodz 90-237 Lodz Poland

5. Chemical biology of ion channels (Chembion) Westfälische Wilhelms-Universität Münster Corrensstraße 48 48149 Münster Germany

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202100735

Reference65 articles.

1. A proposal for the classification of sigma binding sites

2. A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain

3. Rat liver and kidney contain high densities of σ1 and σ2 receptors: characterization by ligand binding and photoaffinity labeling

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