From Quinoline to Quinazoline‐Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search-Reference-Cited by-同舟云学术

From Quinoline to Quinazoline‐Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search

Published:2021-06-26 Issue:19 Volume:16 Page:3044-3059
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Cedraro Nicholas¹,Cannalire Rolando²³^ORCID,Astolfi Andrea³,Mangiaterra Gianmarco¹,Felicetti Tommaso³^ORCID,Vaiasicca Salvatore¹,Cernicchi Giada³,Massari Serena³^ORCID,Manfroni Giuseppe³^ORCID,Tabarrini Oriana³^ORCID,Cecchetti Violetta³^ORCID,Barreca Maria Letizia³^ORCID,Biavasco Francesca¹,Sabatini Stefano³^ORCID

Affiliation:

1. Department of Life and Environmental Sciences Università Politecnica delle Marche via Brecce Bianche 60131 Ancona Italy

2. Current address: Department of Pharmacy University of Napoli “Federico II” via D. Montesano 49 80131 Napoli Italy

3. Department of Pharmaceutical Sciences Università degli Studi di Perugia via del Liceo 1 06123 Perugia Italy

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202100282

Reference56 articles.

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