Stability and Cell Permeability of Sulfonyl Fluorides in the Design of Lys‐Covalent Antagonists of Protein‐Protein Interactions-Reference-Cited by-同舟云学术

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Stability and Cell Permeability of Sulfonyl Fluorides in the Design of Lys‐Covalent Antagonists of Protein‐Protein Interactions

Published:2020-10-13 Issue:22 Volume:15 Page:2176-2184
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Gambini Luca¹,Udompholkul Parima¹,Salem Ahmed F.¹,Baggio Carlo¹,Pellecchia Maurizio¹^ORCID

Affiliation:

1. Biomedical sciences Division School of Medicine University of California Riverside 900 University Avenue CA 92521 Riverside USA

Funder

National Institutes of Health

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202000355

Reference95 articles.

1.

2. Design of Potent pan-IAP and Lys-Covalent XIAP Selective Inhibitors Using a Thermodynamics Driven Approach

3. Covalent Inhibitors of Protein–Protein Interactions Targeting Lysine, Tyrosine, or Histidine Residues

4. Aryl-fluorosulfate-based Lysine Covalent Pan-Inhibitors of Apoptosis Protein (IAP) Antagonists with Cellular Efficacy

5.

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1. De novo design of covalent bonding peptides for target protein;hLife;2024-07

2. Biospecific Chemistry for Covalent Linking of Biomacromolecules;Chemical Reviews;2024-06-24

3. Sulfur (VI) fluoride exchange (SuFEx): a versatile tool to profile protein-biomolecule interactions for therapeutic development;Medicinal Chemistry Research;2024-06-18

4. Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update;Journal of Medicinal Chemistry;2024-05-07

5. Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1;Journal of Medicinal Chemistry;2024-05-02

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