Reproducing prolonged time to peak bisoprolol concentration by PBPK modeling with lysosomal trapping in enterocytes
Author:
Affiliation:
1. Department of Pharmacy Hainan General Hospital (Hainan Affiliated Hospital of Hainan Medical University) Hainan China
2. Clinical Medical College Yangzhou University Yangzhou China
3. Subei People’s Hospital Yangzhou University Yangzhou China
Funder
Natural Science Foundation of Jiangsu Province
Publisher
Wiley
Subject
Pharmacology (medical),Modeling and Simulation
Link
https://onlinelibrary.wiley.com/doi/pdf/10.1002/psp4.12756
Reference5 articles.
1. Application of physiologically based biopharmaceutics modeling to understand the impact of dissolution differences on in vivo performance of immediate release products: The case of bisoprolol
2. Simulation of the pharmacokinetics of bisoprolol in healthy adults and patients with impaired renal function using whole-body physiologically based pharmacokinetic modeling
3. Forecasting oral absorption across biopharmaceutics classification system classes with physiologically based pharmacokinetic models
4. Development and Qualification of Physiologically Based Pharmacokinetic Models for Drugs With Atypical Distribution Behavior: A Desipramine Case Study
5. Early identification of drug-induced impairment of gastric emptying through physiologically based pharmacokinetic (PBPK) simulation of plasma concentration-time profiles in rat
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