Subtype selective fluorescent ligands based on ICI 118,551 to study the human β2‐adrenoceptor in CRISPR/Cas9 genome‐edited HEK293T cells at low expression levels-Reference-Cited by-同舟云学术

Subtype selective fluorescent ligands based on ICI 118,551 to study the human β2‐adrenoceptor in CRISPR/Cas9 genome‐edited HEK293T cells at low expression levels

Published:2021-05 Issue:3 Volume:9 Page:
ISSN:2052-1707
Container-title:Pharmacology Research & Perspectives
language:en
Short-container-title:Pharmacol Res Perspect

Author:

Goulding Joëlle¹²^ORCID,Mistry Sarah J.²³^ORCID,Soave Mark¹²^ORCID,Woolard Jeanette¹²^ORCID,Briddon Stephen J.¹²,White Carl W.¹²⁴⁵^ORCID,Kellam Barrie²³^ORCID,Hill Stephen J.¹²^ORCID

Affiliation:

1. Division of Physiology, Pharmacology and Neuroscience, School of Life Sciences University of Nottingham Nottingham UK

2. Centre of Membrane Proteins and Receptors (COMPARE) University of Birmingham and University of Nottingham Midlands UK

3. School of Pharmacy University of Nottingham Nottingham UK

4. Harry Perkins Institute of Medical Research and Centre for Medical Research University of Western AustraliaQEII Medical Centre Nedlands Western Australia Australia

5. Australian Research Council Centre for Personalised Therapeutics Technologies Australia

Funder

Medical Research Council

Publisher

Wiley

Subject

General Pharmacology, Toxicology and Pharmaceutics,Neurology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/prp2.779

Reference50 articles.

1. International Union of Pharmacology nomenclature of adrenoceptors;Bylund DB;Pharmacol Rev,1994

2. Pharmacology and Therapeutics of Bronchodilators Revisited

3. The β -Adrenoceptor

4. Beta‐adrenergic receptor signaling in cardiac function and heart failure;Madamanchi A;Mcgill J Med,2007

5. NEW INSIGHTS INTO β-ADRENOCEPTORS IN SMOOTH MUSCLE: DISTRIBUTION OF RECEPTOR SUBTYPES and MOLECULAR MECHANISMS TRIGGERING MUSCLE RELAXATION

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Kinetic analysis of fluorescent ligand binding to cell surface receptors: Insights into conformational changes and allosterism in living cells;British Journal of Pharmacology;2023-07-19

2. NanoBiT‐ and NanoBiT/BRET‐based assays allow the analysis of binding kinetics of Wnt‐3a to endogenous Frizzled 7 in a colorectal cancer model;British Journal of Pharmacology;2023-05-06

3. Kinetic analysis of endogenous β ₂ ‐adrenoceptor‐mediated cAMP GloSensor™ responses in HEK293 cells;British Journal of Pharmacology;2023-01-06

4. CELLULAR TARGET ENGAGEMENT ASSAYS FOR SMALL-MOLECULE DRUG DISCOVERY;2022 Medicinal Chemistry Reviews;2022-12-21

5. The use of fluorescence correlation spectroscopy to characterise the molecular mobility of G protein-coupled receptors in membrane microdomains: an update;Biochemical Society Transactions;2021-08-26