High‐Throughput Ligand Screening Enables the Enantioselective Conjugate Borylation of Cyclobutenones to Access Synthetically Versatile Tertiary Cyclobutylboronates-Reference-Cited by-同舟云学术

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High‐Throughput Ligand Screening Enables the Enantioselective Conjugate Borylation of Cyclobutenones to Access Synthetically Versatile Tertiary Cyclobutylboronates

Published:2019-10-31 Issue:51 Volume:131 Page:18576-18580
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Clement Helen A.¹^ORCID,Boghi Michele¹^ORCID,McDonald Rory M.¹^ORCID,Bernier Louise²,Coe Jotham W.³,Farrell William²^ORCID,Helal Christopher J.³^ORCID,Reese Matthew R.³,Sach Neal W.²,Lee Jack C.³,Hall Dennis G.¹^ORCID

Affiliation:

1. Department of Chemistry, 4-010 CCISUniversity of Alberta Edmonton Alberta T6G 2G2 Canada

2. Pfizer Worldwide Research and DevelopmentLa Jolla Laboratories 10770 Science Center Drive San Diego CA 92121 USA

3. Pfizer Worldwide Research and Development Eastern Point Road Groton CT 06340 USA

Funder

Pfizer

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.201909308

Reference51 articles.

1.

2. Naturally occurring bioactive Cyclobutane-containing (CBC) alkaloids in fungi, fungal endophytes, and plants

3. Discovery of Two Clinical Histamine H3 Receptor Antagonists: trans-N-Ethyl-3-fluoro-3-[3-fluoro-4-(pyrrolidinylmethyl)phenyl]cyclobutanecarboxamide (PF-03654746) and trans-3-Fluoro-3-[3-fluoro-4-(pyrrolidin-1-ylmethyl)phenyl]-N-(2-methylpropyl)cyclobutanecarboxamide (PF-03654764)

4. Rigidification:

5. Cyclobutane derivatives as potent NK1 selective antagonists

Cited by 17 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Enantioselective Hydrofunctionalization of Cyclobutenones: Total Synthesis of gem‐Dimethylcyclobutane Natural Products;Angewandte Chemie International Edition;2024-04-11

2. Enantioselective Hydrofunctionalization of Cyclobutenones: Total Synthesis of gem‐Dimethylcyclobutane Natural Products;Angewandte Chemie;2024-04-11

3. Copper-Catalyzed Borylation and Silylation of Dichlorocyclobutenones;Organic Letters;2023-05-08

4. Boosting the Enantioselectivity of Conjugate Borylation of α,β‐Disubstituted Cyclobutenones with Monooxides of Chiral C ₂ ‐Symmetric Bis(phosphine) Ligands;Chemistry – A European Journal;2022-09

5. Stereocontrolled Pericyclic and Radical Cycloaddition Reactions of Readily Accessible Chiral Alkenyl Diazaborolidines;Angewandte Chemie International Edition;2022-06-08

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