Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs-Reference-Cited by-同舟云学术

Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs

Published:2020-01-22 Issue:10 Volume:132 Page:4205-4210
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Dal Corso Alberto¹^ORCID,Borlandelli Valentina¹,Corno Cristina²^ORCID,Perego Paola²^ORCID,Belvisi Laura¹^ORCID,Pignataro Luca¹^ORCID,Gennari Cesare¹^ORCID

Affiliation:

1. Università degli Studi di Milano Dipartimento di Chimica via C. Golgi, 19 20133 Milan Italy

2. Fondazione IRCCS Istituto Nazionale dei Tumori Molecular Pharmacology Unit Department of Applied Research and Technological Development via Amadeo 42 20133 Milan Italy

Funder

Ministero dell’Istruzione, dell’Università e della Ricerca

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.201916394

Reference72 articles.

1. Self-Immolative Spacers: Kinetic Aspects, Structure-Property Relationships, and Applications

2. Selbstzerlegende Spacer: kinetische Aspekte, Struktur-Eigenschafts-Beziehungen und Anwendungen

4. Hmboff/on as a switchable thiol protecting group for native chemical ligation

5. Unprecedented Sensitivity in a Probe for Monitoring Cathepsin B: Chemiluminescence Microscopy Cell-Imaging of a Natively Expressed Enzyme

Cited by 9 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Water-soluble and predictable-release triptolide prodrugs block bleomycin-induced pulmonary fibrosis in mice;European Journal of Medicinal Chemistry;2024-12

2. Amine‐Carbamate Self‐Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads;ChemBioChem;2024-03-14

3. ValCitGlyPro-dexamethasone antibody conjugates selectively suppress the activation of human monocytes;RSC Medicinal Chemistry;2023

4. A Long Journey through Organic Chemistry – Celebrating Cesare Gennari's 70th Birthday;European Journal of Organic Chemistry;2022-11-22

5. Tetrazine‐Triggered Bioorthogonal Cleavage of trans ‐Cyclooctene‐Caged Phenols Using a Minimal Self‐Immolative Linker Strategy**;ChemBioChem;2022-08-30