Selective α-Monomethylation by an Amine-Borane/N ,N -Dimethylformamide System as the Methyl Source-Reference-Cited by-同舟云学术

Selective α-Monomethylation by an Amine-Borane/N ,N -Dimethylformamide System as the Methyl Source

Published:2018-08-01 Issue:36 Volume:130 Page:11944-11949
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Xia Hui-Min¹,Zhang Feng-Lian¹,Ye Tian¹,Wang Yi-Feng¹²^ORCID

Affiliation:

1. Hefei National Laboratory for Physical Sciences at the Microscale; Center for Excellence in Molecular Synthesis of CAS, and; Department of Chemistry; University of Science and Technology of China; 96 Jinzhai Road Hefei Anhui 230026 China

2. State Key Laboratory of Elemento-Organic Chemistry; Nankai University; Tianjin 300071 China

Funder

University of Science and Technology of China

National Natural Science Foundation of China

Fundamental Research Funds for the Central Universities

Recruitment Program of Global Experts

China Postdoctoral Science Foundation

Publisher

Wiley

Subject

General Medicine

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/ange.201804794/fullpdf

Reference83 articles.

1. Profound Methyl Effects in Drug Discovery and a Call for New CH Methylation Reactions

2. Ausgeprägte Methyleffekte in der Wirkstoff-Forschung und der Bedarf an neuen C-H-Methylierungsreaktionen

3. The Methylation Effect in Medicinal Chemistry

4. Methyl Effects on Protein–Ligand Binding

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