Selectivity in the impact of P-glycoprotein upon pulmonary absorption of airway-dosed substrates: A study in ex vivo lung models using chemical inhibition and genetic knockout
Author:
Publisher
Elsevier BV
Subject
Pharmaceutical Science
Reference40 articles.
1. Spatial expression and functionality of drug transporters in the intact lung: Objectives for further research;Gumbleton;Adv Drug Deliv Rev,2011
2. Drug transporters in the lung—Do they play a role in the biopharmaceutics of inhaled drugs?;Bosquillon;J Pharm Sci,2010
3. Organic cation transporters in the blood-air barrier: Expression and implications for pulmonary drug delivery;Salomon;Ther Deliv,2012
4. Constitutive expression of P-glycoprotein in normal lung alveolar epithelium and functionality in primary alveolar epithelial cultures;Campbell;J Pharmacol Exp Ther,2003
5. Tissue distribution and chemical induction of multiple drug resistance genes in rats;Brady;Drug Metab Dispos,2002
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