Second-Generation Inhibitors for the Metalloprotease Neprilysin Based on Bicyclic Heteroaromatic Scaffolds: Synthesis, Biological Activity, and X-Ray Crystal-Structure Analysis-Reference-Cited by-同舟云学术

Second-Generation Inhibitors for the Metalloprotease Neprilysin Based on Bicyclic Heteroaromatic Scaffolds: Synthesis, Biological Activity, and X-Ray Crystal-Structure Analysis

Published:2005-04 Issue:4 Volume:88 Page:731-750
ISSN:0018-019X
Container-title:Helvetica Chimica Acta
language:en
Short-container-title:HCA

Author:

Sahli Stefan,Frank Brian,Schweizer W. Bernd,Diederich François,Blum-Kaelin Denise,Aebi Johannes D.,Böhm Hans-Joachim,Oefner Christian,Dale Glenn E.

Publisher

Wiley

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery,Biochemistry,Catalysis

Reference42 articles.

1. A New Class of Inhibitors for the Metalloprotease Neprilysin Based on a Central Imidazole Scaffold

2. Structure of human neutral endopeptidase (neprilysin) complexed with phosphoramidon 1 1Edited by R. Huber

3. The enkephalinase inhibitor thiorphan shows antinociceptive activity in mice

4. Three-Dimensional Models of ACE and NEP Inhibitors and Their Use in the Design of Potent Dual ACE/NEP Inhibitors

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