Design, Synthesis and in vitro Evaluation of Indolotacrine Analogues as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease

Author:

Benek Ondrej123,Soukup Ondrej23,Pasdiorova Marketa13,Hroch Lukas34,Sepsova Vendula13,Jost Petr13,Hrabinova Martina13,Jun Daniel1,Kuca Kamil35,Zala Dominykas6,Ramsay Rona R.6,Marco-Contelles José7,Musilek Kamil35

Affiliation:

1. Department of Toxicology and Military Pharmacy; Department of Epidemiology, Faculty of Military Health Sciences; University of Defense; Trebesska 1575 500 01 Hradec Kralove Czech Republic

2. National Institute of Mental Health; Topolova 748 250 67 Klecany Czech Republic

3. University Hospital; Sokolska 581 500 05 Hradec Kralove Czech Republic

4. Department of Pharmaceutical Chemistry and Drug Control; Faculty of Pharmacy in Hradec Kralove; Charles University in Prague; Akademika Heyrovskeho 1203 500 05 Hradec Kralove Czech Republic

5. Department of Chemistry; Faculty of Science; University of Hradec Kralove; Rokitanskeho 62 500 03 Hradec Kralove Czech Republic

6. School of Biology, Biomolecular Sciences Building; University of St. Andrews; North Haugh St. Andrews KY16 9ST UK

7. Laboratory of Medicinal Chemistry; (IQOG, CSIC); Juan de la Cierva 3 28006 Madrid Spain

Funder

Czech National Institute of Mental Health (NIMH-CZ)

Ministry of Education, Youth and Sports of the Czech Republic

MH CZ-DRO

UHHK

University of Defense of the Czech Republic

MINECO

Government of Spain

School of Biology at the University of St. Andrews

COST Action

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

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