Development of submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation-Reference-Cited by-同舟云学术

Development of submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation

Published:2023-10 Issue: Volume:258 Page:115593
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Benek Ondrej^ORCID,Vaskova Michaela,Miskerikova Marketa,Schmidt Monika,Andrys Rudolf,Rotterova Aneta,Skarka Adam,Hatlapatkova Jana,Karasova Jana Zdarova,Medvecky Matej,Hroch Lukas,Vinklarova Lucie,Fisar Zdenek,Hroudova Jana,Handl Jiri,Capek Jan,Rousar Tomas,Kobrlova Tereza,Dolezal Rafael,Soukup Ondrej,Aitken Laura,Gunn-Moore Frank,Musilek Kamil^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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1. C-3 Steroidal Hemiesters as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 10;ACS Omega;2024-02-28

2. Involvement of Type 10 17β-Hydroxysteroid Dehydrogenase in the Pathogenesis of Infantile Neurodegeneration and Alzheimer’s Disease;International Journal of Molecular Sciences;2023-12-18

3. Nanomolar Benzothiazole-Based Inhibitors of 17β-HSD10 with Cellular Bioactivity;ACS Medicinal Chemistry Letters;2023-11-10

4. Physiologically relevant fluorescent assay for identification of 17β‐hydroxysteroid dehydrogenase type 10 inhibitors;Journal of Neurochemistry;2023-07-17