Synthesis and Structure‐Activity Relationships of N ‐(4‐Benzamidino)‐Oxazolidinones: Potent and Selective Inhibitors of Kallikrein‐Related Peptidase 6-Reference-Cited by-同舟云学术

Synthesis and Structure‐Activity Relationships of N ‐(4‐Benzamidino)‐Oxazolidinones: Potent and Selective Inhibitors of Kallikrein‐Related Peptidase 6

Published:2019-11-18 Issue:1 Volume:15 Page:79-95
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

De Vita Elena¹²^ORCID,Smits Niels³,Hurk Helma³,Beck Elizabeth M.⁴,Hewitt Joanne⁴,Baillie Gemma⁴,Russell Emily⁴,Pannifer Andrew⁴,Hamon Véronique⁴,Morrison Angus⁴,McElroy Stuart P.⁴,Jones Philip⁴,Ignatenko Natalia A.⁵⁶,Gunkel Nikolas¹⁷,Miller Aubry K.¹⁷^ORCID

Affiliation:

1. Cancer Drug Development GroupGerman Cancer Research Center (DKFZ) Im Neuenheimer Feld 280 69120 Heidelberg Germany

2. Faculty of BiosciencesUniversity of Heidelberg 69120 Heidelberg Germany

3. Pivot Park Screening Centre Kloosterstraat 9 5349 AB Oss (The Netherlands

4. European Screening Centre Newhouse (ESC) Biocity Scotland Bo'ness Road ML15UH Newhouse Scotland

5. University of Arizona Cancer CenterUniversity of Arizona Tucson AZ 85721 USA

6. Department of Cellular and Molecular MedicineUniversity of Arizona Tucson AZ 85721 USA

7. German Cancer Consortium (DKTK) 69120 Heidelberg Germany

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201900536

Reference39 articles.

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