Controlling the Covalent Reactivity of a Kinase Inhibitor with Light-Reference-Cited by-同舟云学术

Controlling the Covalent Reactivity of a Kinase Inhibitor with Light

Published:2021-08-11 Issue:37 Volume:133 Page:20340-20345
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Reynders Martin¹²^ORCID,Chaikuad Apirat³⁴⁵^ORCID,Berger Benedict‐Tilman³⁴⁵^ORCID,Bauer Katharina⁶⁷,Koch Pierre⁶⁷⁸^ORCID,Laufer Stefan⁶⁷^ORCID,Knapp Stefan³⁴⁵⁹^ORCID,Trauner Dirk¹^ORCID

Affiliation:

1. Department of Chemistry, Silver Center for Arts and Science New York University 100 Washington Square East New York NY 10003 USA

2. Department of Chemistry Ludwig Maximilians University of Munich Butenandtstr.5–13 81377 Munich Germany

3. Buchmann Institute for Molecular Life Sciences Johann Wolfgang Goethe-University 60438 Frankfurt am Main Germany

4. Institute for Pharmaceutical Chemistry Johann Wolfgang Goethe-University 60438 Frankfurt am Main Germany

5. Structural Genomics Consortium Frankfurt 60438 Frankfurt am Main Germany

6. Department of Pharmaceutical/ Medicinal Chemistry Eberhard-Karls-University Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany

7. Tuebingen Center for Academic Drug Discovery Germany

8. Department of Pharmaceutical/Medicinal Chemistry II Institute of Pharmacy University of Regensburg 93040 Regensburg Germany

9. German Cancer Network (DKTK) Frankfurt/Mainz site 60438 Frankfurt am Main Germany

Funder

National Institutes of Health

Deutsche Forschungsgemeinschaft

German Cancer Research Center

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.202103767

Reference33 articles.

1. Properties of FDA-approved small molecule protein kinase inhibitors

2. Developing Irreversible Inhibitors of the Protein Kinase Cysteinome

3. The Cysteinome of Protein Kinases as a Target in Drug Development

4. Das Cysteinom der Proteinkinasen als Zielstruktur in der Arzneistoffentwicklung

5. On‐Command Regulation of Kinase Activity using Photonic Stimuli

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