Potent Trivalent Inhibitors of Thrombin through Hybridization of Salivary Sulfopeptides from Hematophagous Arthropods-Reference-Cited by-同舟云学术

Potent Trivalent Inhibitors of Thrombin through Hybridization of Salivary Sulfopeptides from Hematophagous Arthropods

Published:2021-01-28 Issue:10 Volume:133 Page:5408-5416
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Agten Stijn M.¹²^ORCID,Watson Emma E.¹^ORCID,Ripoll‐Rozada Jorge³^ORCID,Dowman Luke J.¹^ORCID,Wu Mike C. L.⁴⁵^ORCID,Alwis Imala⁴⁵^ORCID,Jackson Shaun P.⁴⁵^ORCID,Pereira Pedro José Barbosa³^ORCID,Payne Richard J.¹^ORCID

Affiliation:

1. School of Chemistry and ARC Centre of Excellence for Innovations in Peptide and Protein Science The University of Sydney Sydney NSW 2006 Australia

2. Department of Biochemistry, Cardiovascular Research Institute Maastricht (CARIM) Maastricht University Universiteitssingel 50 6229 ER Maastricht The Netherlands

3. IBMC—Instituto de Biologia Molecular e Celular and Instituto de Investigação e Inovação em Saúde Universidade do Porto 4200-135 Porto Portugal

4. Charles Perkins Centre The University of Sydney Sydney NSW 2006 Australia

5. Heart Research Institute Sydney NSW 2042 Australia

Funder

National Health and Medical Research Council

CARIM School for Cardiovascular Diseases, Universiteit Maastricht

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.202015127

Reference35 articles.

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2. A player of many parts: The spotlight falls on thrombin's structure

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4. The Structure of a Complex of Recombinant Hirudin and Human α-Thrombin

5. Variegin, a Novel Fast and Tight Binding Thrombin Inhibitor from the Tropical Bont Tick