Synthesis and evaluation of novel 4 H ‐pyrazole and thiophene derivatives derived from chalcone as potential anti‐proliferative agents, Pim‐1 kinase inhibitors, and PAINS-Reference-Cited by-同舟云学术

Synthesis and evaluation of novel 4 H ‐pyrazole and thiophene derivatives derived from chalcone as potential anti‐proliferative agents, Pim‐1 kinase inhibitors, and PAINS

Published:2020-04 Issue:4 Volume:57 Page:1993-2009
ISSN:0022-152X
Container-title:Journal of Heterocyclic Chemistry
language:en
Short-container-title:J Heterocycl Chem

Author:

Megally Abdo Nadia Y.¹^ORCID,Samir Eman M.²,Mohareb Rafat M.³^ORCID

Affiliation:

1. Chemistry Department, Faculty of EducationAlexandria University Alexandria A. R. Egypt

2. Department of Organic Chemistry, National Organization for Drug Control & Research (NODCAR), P.O. 29 Cairo A. R. Egypt

3. Department of Chemistry, Faculty of ScienceCairo University Cairo A. R. Egypt

Publisher

Wiley

Subject

Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/jhet.3928

Reference61 articles.

1. A review of anti-infective and anti-inflammatory chalcones

2. Practical Synthesis of Chalcone Derivatives and Their Biological Activities

3. Synthesis, Characterization, Antimicrobial Screening and Free-Radical Scavenging Activity of Some Novel Substituted Pyrazoles

4. Application of chalcones in heterocycles synthesis: Synthesis of 2-(isoxazolo, pyrazolo and pyrimido) substituted analogues of 1,4-benzodiazepin-5-carboxamides linked through an oxyphenyl bridge

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