Donepezil-melatonin hybrids as butyrylcholinesterase inhibitors: Improving binding affinity through varying mode of linking fragments-Reference-Cited by-同舟云学术

Donepezil-melatonin hybrids as butyrylcholinesterase inhibitors: Improving binding affinity through varying mode of linking fragments

Published:2018-10-05 Issue:11 Volume:351 Page:1800194
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Arch. Pharm. Chem. Life Sci.

Author:

Łozińska Iwona¹,Świerczyńska Aleksandra¹,Molęda Zuzanna¹^ORCID,Hartman Alwin M.²^ORCID,Hirsch Anna K. H.²³^ORCID,Czarnocki Zbigniew¹^ORCID

Affiliation:

1. Faculty of Chemistry; University of Warsaw; Warsaw Poland

2. Department of Drug Design and Optimization; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS) - Helmholtz Centre for Infection Research (HZI); Saarbrücken Germany

3. Department of Pharmacy, Medicinal Chemistry; Saarland University; Saarbrücken Germany

Funder

Helmholtz-Association's Initiative and Networking Fund

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/ardp.201800194/fullpdf

Reference29 articles.

1. Acetylcholinesterase Inhibitors: Pharmacology and Toxicology

2. Butyrylcholinesterase-knockout reduces brain deposition of fibrillar β-amyloid in an Alzheimer mouse model

3. Review of human butyrylcholinesterase structure, function, genetic variants, history of use in the clinic, and potential therapeutic uses

4. Selective butyrylcholinesterase inhibition elevates brain acetylcholine, augments learning and lowers Alzheimer -amyloid peptide in rodent

5. Recent progress in the identification of selective butyrylcholinesterase inhibitors for Alzheimer's disease

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