New Tripeptide-Based Macrocyclic Calpain Inhibitors Formed byN-Alkylation of Histidine-Reference-Cited by-同舟云学术

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New Tripeptide-Based Macrocyclic Calpain Inhibitors Formed byN-Alkylation of Histidine

Published:2012-11 Issue:11 Volume:9 Page:2473-2484
ISSN:1612-1872
Container-title:Chemistry & Biodiversity
language:en
Short-container-title:Chemistry & Biodiversity

Author:

Chen Hongyuan,Jiao Wanting,Jones Matthew A.,Coxon James M.,Morton James D.,Bickerstaffe Roy,Pehere Ashok D.,Zvarec Ondrej,Abell Andrew D.

Publisher

Wiley

Subject

Molecular Biology,Molecular Medicine,General Chemistry,Biochemistry,General Medicine,Bioengineering

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cbdv.201200320/fullpdf

Reference30 articles.

1. Molecular Modeling, Synthesis, and Biological Evaluation of Macrocyclic Calpain Inhibitors

2. New β-Strand Templates Constrained by Huisgen Cycloaddition

3. Conformational Selection of Inhibitors and Substrates by Proteolytic Enzymes: Implications for Drug Design and Polypeptide Processing

4. Countering Cooperative Effects in Protease Inhibitors Using Constrained β-Strand-Mimicking Templates in Focused Combinatorial Libraries

5. β-Strand Mimicking Macrocyclic Amino Acids: Templates for Protease Inhibitors with Antiviral Activity

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1. Mechanism-Based Macrocyclic Inhibitors of Serine Proteases;Journal of Medicinal Chemistry;2024-03-13

2. Design, synthesis, and applications of ring‐functionalized histidines in peptide‐based medicinal chemistry and drug discovery;Medicinal Research Reviews;2023-01-29

3. Cyclisation strategies for stabilising peptides with irregular conformations;RSC Medicinal Chemistry;2021

4. Modulators of calpain activity: inhibitors and activators as potential drugs;Expert Opinion on Drug Discovery;2020-02-05

5. An efficient green diversity oriented synthesis of pyrimidinone and indole appended macrocyclic peptidomimetics;Tetrahedron Letters;2019-01

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