Petasis/Diels-Alder/Cyclization Cascade Reactions for the Generation of Scaffolds with Multiple Stereogenic Centers and Orthogonal Handles for Library Production-Reference-Cited by-同舟云学术

Petasis/Diels-Alder/Cyclization Cascade Reactions for the Generation of Scaffolds with Multiple Stereogenic Centers and Orthogonal Handles for Library Production

Published:2018-06-15 Issue:36 Volume:2018 Page:5023-5029
ISSN:1434-193X
Container-title:European Journal of Organic Chemistry
language:en
Short-container-title:Eur. J. Org. Chem.

Author:

Flagstad Thomas¹²,Azevedo Carlos M. G.¹²,Min Geanna¹²,Willaume Anthony³,Morgentin Rémy³,Nielsen Thomas E.¹⁴⁵,Clausen Mads H.¹²^ORCID

Affiliation:

1. Department of Chemistry; Technical University of Denmark; 2800 Kgs. Lyngby Denmark

2. Center for Nanomedicine and Theranostics; Technical University of Denmark; 2800 Kgs. Lyngby Denmark

3. EDELRIS; 115 Avenue Lacassagne 69003 Lyon France

4. Singapore Centre on Environmental Life Science Engineering; Nanyang Technological University; 637551 Singapore Singapore

5. Costerton Biofilm Center; Department of Immunology and Microbiology; University of Copenhagen; 2200 Copenhagen DK- Denmark

Funder

FP7 Ideas: European Research Council

Publisher

Wiley

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/ejoc.201800565/fullpdf

Reference19 articles.

1. 2017 FDA drug approvals

2. What Do Medicinal Chemists Actually Make? A 50-Year Retrospective

3. Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

4. Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?

5. The impact of aromatic ring count on compound developability: further insights by examining carbo- and hetero-aromatic and -aliphatic ring types

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