Synthesis and biological evaluation of novel NK-1 tachykinin receptor antagonists: The use of cycloalkyl amino acids as a template-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of novel NK-1 tachykinin receptor antagonists: The use of cycloalkyl amino acids as a template

Published:1995-10 Issue:4 Volume:36 Page:511-524
ISSN:0006-3525
Container-title:Biopolymers
language:en
Short-container-title:Biopolymers

Author:

Sisto Alessandro,Bonelli Fabio,Centini Felice,Fincham Christopher I.,Potier Edoardo,Monteagudo Edith,Lombardi Paolo,Arcamone Federico,Goso Cristina,Manzini Stefano,Giolitti Alessandro,Maggi Carlo A.,Venanzi Mariano,Pispisa Basilio

Publisher

Wiley

Subject

Organic Chemistry,Biomaterials,Biochemistry,General Medicine,Biophysics

Reference31 articles.

1. Tachykinin receptors and tachykinin receptor antagonists

2. Intraneuronal Substance P Contributes to the Severity of Experimental Arthritis

3. Receptor binding sites for substance P, but not substance K or neuromedin K, are expressed in high concentrations by arterioles, venules, and lymph nodules in surgical specimens obtained from patients with ulcerative colitis and Crohn disease.

4. Studies on neurokinin antagonists. 2. Design and structure-activity relationships of novel tripeptide substance P antagonists, N.alpha.-[N.alpha.-(N.alpha.-acetyl-L-threonyl)-N1-formyl-D-tryptophyl]-N-methyl-N-(phenylmethyl)-L-phenylalaninamide and its related compounds

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