Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents-Reference-Cited by-同舟云学术

Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents

Published:2015-04-17 Issue:3 Volume:4 Page:342-362
ISSN:2191-1363
Container-title:ChemistryOpen
language:en
Short-container-title:ChemistryOpen

Author:

Russo Francesco¹,Gising Johan¹,Åkerbladh Linda¹,Roos Annette K.²,Naworyta Agata³,Mowbray Sherry L.²,Sokolowski Anders¹,Henderson Ian⁴,Alling Torey⁵,Bailey Mai A.⁵,Files Megan⁵,Parish Tanya⁵,Karlén Anders¹,Larhed Mats⁶

Affiliation:

1. Department of Medicinal Chemistry; Organic Pharmaceutical Chemistry, BMC; Uppsala University; Box 574 751 23 Uppsala Sweden

2. Department of Cell and Molecular Biology; Science for Life Laboratory, BMC; Uppsala University; Box 596 751 24 Uppsala Sweden

3. Department of Cell and Molecular Biology, BMC; Uppsala University; Box 596 751 24 Uppsala Sweden

4. Medivir AB; PO Box 1086 141 22 Huddinge Sweden

5. TB Discovery Research; Infectious Disease Research Institute; Seattle WA 98102 USA

6. Department of Medicinal Chemistry; Science for Life Laboratory, BMC; Uppsala University; Box 574 751 23 Uppsala Sweden

Funder

VINNOVA-the Swedish Governmental Agency for Innovation Systems

Bill and Melinda Gates Foundation

National Institute of Allergy and Infectious Diseases (NIAID) of the National Institutes of Health

National Institutes of Health

Publisher

Wiley

Subject

General Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/open.201500001/fullpdf

Reference61 articles.

1. 2014

2. Totally Drug-Resistant Tuberculosis in India

3. Emergence of New Forms of Totally Drug-Resistant Tuberculosis Bacilli

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