Inhibition of Human DHODH by 4-Hydroxycoumarins, Fenamic Acids, andN-(Alkylcarbonyl)anthranilic Acids Identified by Structure-Guided Fragment Selection-Reference-Cited by-同舟云学术

Inhibition of Human DHODH by 4-Hydroxycoumarins, Fenamic Acids, andN-(Alkylcarbonyl)anthranilic Acids Identified by Structure-Guided Fragment Selection

Published:2010-04-06 Issue:4 Volume:5 Page:608-617
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Fritzson Ingela,Svensson Bo,Al-Karadaghi Salam,Walse Björn,Wellmar Ulf,Nilsson Ulf J.,da Graça Thrige Dorthe,Jönsson Stig

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.200900454/fullpdf

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1. T-lymphocytes from AIDS Patients Are Unable to Synthesize Ribonucleotides de Novo in Response to Mitogenic Stimulation

2. Inhibitors of dihydroorotate dehydrogenase

3. Multicenter phase II study of brequinar sodium in patients with advanced lung cancer

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