Nano‐in‐Microparticles for Aerosol Delivery of Antibiotic‐Loaded, Fucose‐Derivatized, and Macrophage‐Targeted Liposomes to Combat Mycobacterial Infections: In Vitro Deposition, Pulmonary Barrier Interactions, and Targeted Delivery

Author:

Huck Benedikt C.12,Thiyagarajan Durairaj3,Bali Aghiad12,Boese Annette1,Besecke Karen F. W.4,Hozsa Constantin4,Gieseler Robert K.45,Furch Marcus4,Carvalho‐Wodarz Cristiane1,Waldow Franziska67,Schwudke Dominik678,Metelkina Olga910,Titz Alexander91011,Huwer Hanno12,Schwarzkopf Konrad13,Hoppstädter Jessica14,Kiemer Alexandra K.14,Koch Marcus15,Loretz Brigitta1ORCID,Lehr Claus‐Michael12ORCID

Affiliation:

1. Department of Drug Delivery Helmholtz Institute for Pharmaceutical Research Saarland Campus E8.1 Saarbrücken 66123 Germany

2. Department of Pharmacy Helmholtz Institute for Pharmaceutical Research Saarland Saarland University Campus E8 1 Saarbrücken 66123 Germany

3. Department of Anti‐infective Drug Discovery Helmholtz Institute for Pharmaceutical Research Saarland Campus E8 1 Saarbrücken 66123 Germany

4. Rodos Biotarget GmbH Hannover 30625 Germany

5. Laboratory of Immunology and Molecular Biology and Department of Internal Medicine University Hospital Knappschaftskrankenhaus Bochum Ruhr University Bochum Bochum 44892 Germany

6. Research Center Borstel Leibniz Lung Center Borstel 23845 Germany

7. German Center for Infection Research Thematic Translational Unit Tuberculosis Partner Site Hamburg‐Lübeck‐Borstel‐Riems Braunschweig 38124 Germany

8. German Center for Lung Research (DZL) Airway Research Center North (ARCN) Kiel Nano Surface and Interface Science KiNSIS Kiel University Kiel 24118 Germany

9. Chemical Biology of Carbohydrates (CBCH) Helmholtz‐Institute for Pharmaceutical Research Saarland (HIPS) Helmholtz Center for Infection Research Saarbrücken 66123 Germany

10. Department of Chemistry Saarland University Saarbrücken 66123 Germany

11. Deutsches Zentrum für Infektionsforschung (DZIF) Hannover‐Braunschweig site Braunschweig 38124 Germany

12. Cardiothoracic Surgery Heart Center Voelklingen Völklingen 66333 Germany

13. Department of Anaesthesia and Intensive Care Klinikum Saarbrücken gGmbH Saarbrücken 66119 Germany

14. Pharmaceutical Biology Saarland University Campus C2 3 Saarbrücken 66123 Germany

15. INM – Leibniz Institute for New Materials Campus D2 2 Saarbrücken 66123 Germany

Publisher

Wiley

Subject

Pharmaceutical Science,Biomedical Engineering,Biomaterials

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