Discovery of New Phosphoinositide 3-kinase Delta (PI3Kδ) Inhibitors via Virtual Screening using Crystallography-derived Pharmacophore Modelling and QSAR Analysis
Author:
Affiliation:
1. Faculty of Pharmacy, Zarqa University, P.O. Box 132222, Zarqa, 13132, Jordan
2. Department of Pharmaceutical Sciences, Faculty of Pharmacy, The University of Jordan, Amman, Jordan
Abstract
Funder
Zarqa University
Publisher
Bentham Science Publishers Ltd.
Subject
Drug Discovery
Reference86 articles.
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3. Study results provide rationale for use of PI3K inhibitors in therapeutic settings, News-medical.net. Retrieved on 2010-11-0
4. Crabbe T.; Exploring the potential of PI3K inhibitors for inflammation and cancer. Biochem Soc Trans 2007,35(Pt 2),253-256
5. Stein R.; Prospects for phosphoinositide 3-kinase inhibition as a cancer treatment”. Endocr. Relat. Cancer. Bioscientifica 2001,8(3),237-348
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