Development of phosphoinositide 3-kinase delta (PI3Kδ) inhibitors as potential anticancer agents through the generation of ligand-based pharmacophores and biological screening
Author:
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
https://link.springer.com/content/pdf/10.1007/s00044-023-03057-3.pdf
Reference60 articles.
1. Janku F. Phosphoinositide 3-kinase (PI3K) pathway inhibitors in solid tumors: from laboratory to patients. Cancer Treat Rev. 2017;59:93–101. https://doi.org/10.1016/j.ctrv.2017.07.005.
2. Ito K, Caramori G, Adcock IM. Therapeutic potential of phosphatidylinositol 3-kinase inhibitors in inflammatory respiratory disease. Pharmacol Exp Ther. 2007;321:1–8. https://doi.org/10.1124/jpet.106.111674.
3. Du J, Yang M, Chen S, Li D, Chang Z, Dong Z. PDK1 promotes tumor growth and metastasis in a spontaneous breast cancer model. Oncogene. 2016;35:3314–23. https://doi.org/10.1038/onc.2015.393.
4. Crabbe T. Exploring the potential of PI3K inhibitors for inflammation and cancer. Biochem Soc Trans. 2007;35:253–6. https://doi.org/10.1042/bst0350253.
5. Stein RC. Prospects for phosphoinositide 3-kinase inhibition as a cancer treatment. Endocr-Relat Cancer. 2001;8:237–48. https://doi.org/10.1677/erc.0.0080237.
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