Nitrogen-containing Heterocycle: A Privileged Scaffold for Marketed Drugs
Author:
Affiliation:
1. Henan Provincial Key Laboratory Of Children's Genetics and Metabolic Diseases, Children's Hospital Affiliated to Zhengzhou University, Zhengzhou Children's Hospital, Zhengzhou University, Zhengzhou 450018,China
Abstract
Funder
China Postdoctoral Science Foundation
Postdoctoral Research Grant in Henan Province
Henan Medical Science and Technology Program
Publisher
Bentham Science Publishers Ltd.
Subject
Drug Discovery,General Medicine
Reference10 articles.
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3. Pennington L.D.; Moustakas D.T.; The necessary nitrogen atom: a versatile high-impact design element for multiparameter optimization. J Med Chem 2017,60(9),3552-3579
4. Duan Y.; Liu W.; Tian L.; Mao Y.; Song C.; Targeting tubulin-colchicine site for cancer therapy: inhibitors, antibody- drug conjugates and degradation agents. Curr Top Med Chem 2019,19(15),1289-1304
5. Wang Y.; Yao Y.; Zhu H.L.; Duan Y.; Butterfly structure: a privileged scaffold targeting tubulin-colchicine binding site. Curr Top Med Chem 2020,20(17),1505-1508
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