Pharmacokinetics of ruboxistaurin are significantly altered by rifampicin-mediated CYP3A4 induction
Author:
Publisher
Wiley
Subject
Pharmacology (medical),Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1365-2125.2005.02540.x/fullpdf
Reference36 articles.
1. 1MR Jirousek, JR Gillig, CM Gonzalez, WF Heath, JH McDonald, DA rd. Neel, CJ Rito, U Singh, LE Stramm, A Melikian-Badalian, M Baevsky, LM Ballas, SE Hall, LL Winneroski, MM. Faul, andbv(S)-13-[(Dimethylamino) methyl]-10,11,14,15-tetrahydro-4,9: 16,21-dimetheno-1H,13H-dibenzo[e,k]pyrrolo[3,4-h][1,4,13] oxadiazacyclohexadecene-1,3 (2H)-dione (ruboxistaurin) and related analogues: Isozyme selective inhibitors of protein kinase C beta . J Med Chem1996 : 39:2664-71.
2. The Potential Role of PKC β in Diabetic Retinopathy and Macular Edema
3. A novel potential therapy for diabetic nephropathy and vascular complications: protein kinase C β inhibition
4. Salt form selection and characterization of LY333531 mesylate monohydrate
5. Elevated glucose promotes generation of endothelium-derived vasoconstrictor prostanoids in rabbit aorta.
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