Human microdose evaluation of the novel EP1 receptor antagonist GSK269984A
Author:
Publisher
Wiley
Subject
Pharmacology (medical),Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1365-2125.2012.04296.x/fullpdf
Reference53 articles.
1. Prostaglandin E receptors;Sugimoto;J Biol Chem,2007
2. Reduced pain hypersensitivity and inflammation in mice lacking microsomal prostaglandin e synthase-1;Kamei;J Biol Chem,2004
3. Impaired inflammatory and pain responses in mice lacking an inducible prostaglandin E synthase;Trebino;Proc Natl Acad Sci U S A,2003
4. Microsomal prostaglandin E2 synthase-1 (mPGES-1): a novel anti-inflammatory therapeutic target;Friesen;J Med Chem,2008
5. MF63 [2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)-isophthalonitrile], a selective microsomal prostaglandin E synthase-1 inhibitor, relieves pyresis and pain in preclinical models of inflammation;Xu;J Pharmacol Exp Ther,2008
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