Pharmacodynamics, pharmacokinetics and safety of GSK2190915, a novel oral anti-inflammatory 5-lipoxygenase-activating protein inhibitor-Reference-Cited by-同舟云学术

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Pharmacodynamics, pharmacokinetics and safety of GSK2190915, a novel oral anti-inflammatory 5-lipoxygenase-activating protein inhibitor

Published:2013-02-05 Issue:3 Volume:75 Page:779-790
ISSN:0306-5251
Container-title:British Journal of Clinical Pharmacology
language:en
Short-container-title:Br J Clin Pharmacol

Author:

Bain Gretchen¹,King Christopher D.¹,Schaab Kevin,Rewolinski Melissa²,Norris Virginia³,Ambery Claire³,Bentley Jane³,Yamada Masanori⁴,Santini Angelina M.¹,van de Wetering de Rooij Jeroen⁵,Stock Nicholas⁶,Zunic Jasmine,Hutchinson John H.⁷,Evans Jilly F.

Affiliation:

1. Bristol-Myers Squibb; San Diego CA USA

2. Intercept Pharmaceuticals; San Diego CA USA

3. GSK; Stevenage UK

4. GSK; Tokyo Japan

5. PRA International Group B.V.; Zuidlaren the Netherlands

6. Inception Sciences; San Diego CA

7. Brain Cells, Inc; San Diego CA USA

Funder

Amira Pharmaceuticals, Inc.

GlaxoSmithKline (GSK)

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1365-2125.2012.04386.x/fullpdf

Reference27 articles.

1. The nuclear membrane organization of leukotriene synthesis;Mandal;Proc Natl Acad Sci U S A,2008

2. Identification and isolation of a membrane protein necessary for leukotriene production;Miller;Nature,1990

3. Leukotriene signaling in atherosclerosis and ischemia;Back;Cardiovasc Drugs Ther,2009

4. The gene encoding 5-lipoxygenase activating protein confers risk of myocardial infarction and stroke;Helgadottir;Nat Genet,2004

5. The role of LTA4H and ALOX5AP polymorphism in asthma and allergy susceptibility;Holloway;Allergy,2008

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2. Novel Chemical Series of 5-Lipoxygenase-Activating Protein Inhibitors for Treatment of Coronary Artery Disease;Journal of Medicinal Chemistry;2019-03-30

3. Novel leukotriene biosynthesis inhibitors (2012-2016) as anti-inflammatory agents;Expert Opinion on Therapeutic Patents;2017-01-05

4. BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly;Biochemical Pharmacology;2016-11

5. Novel approaches to the management of noneosinophilic asthma;Therapeutic Advances in Respiratory Disease;2016-02-28

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