Crystal Structures of IL-2-inducible T cell Kinase Complexed with Inhibitors: Insights into Rational Drug Design and Activity Regulation-Reference-Cited by-同舟云学术

Crystal Structures of IL-2-inducible T cell Kinase Complexed with Inhibitors: Insights into Rational Drug Design and Activity Regulation

Published:2010-06-09 Issue:2 Volume:76 Page:154-163
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:

Author:

Kutach Alan K.,Villaseñor Armando G.,Lam Diana,Belunis Charles,Janson Cheryl,Lok Stephen,Hong Li-Na,Liu Chao-Min,Deval Jerome,Novak Thomas J.,Barnett Jim W.,Chu Wei,Shaw David,Kuglstatter Andreas

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Reference35 articles.

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4. Mechanism and functional significance of Itk autophosphorylation;Joseph;J Mol Biol,2007

5. The linker between SH2 and kinase domains positively regulates catalysis of the Tec family kinases;Joseph;Biochemistry,2007

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