Pharmacological profile of opicapone, a third-generation nitrocatechol catechol-O-methyl transferase inhibitor, in the rat
Author:
Affiliation:
1. Department of Research and Development; BIAL - Portela & Cª, S.A.; São Mamede do Coronado Portugal
2. Department of Pharmacology and Therapeutics; Faculty of Medicine; University of Porto; Porto Portugal
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/bph.13020/fullpdf
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3. Kinetic inhibitory profile of BIA 3-202, a novel fast tight-binding, reversible and competitive catechol-O-methyltransferase inhibitor;Bonifácio;Eur J Pharmacol,2003
4. Catechol-O-methyltransferase and its inhibitors in Parkinson's disease;Bonifácio;CNS Drug Rev,2007
5. Brain and peripheral pharmacokinetics of levodopa in the cynomolgus monkey following administration of opicapone, a third generation nitrocatechol COMT inhibitor;Bonifácio;Neuropharmacology,2014
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