Structure‐based discovery of ( S )‐2‐amino‐6‐(4‐fluorobenzyl)‐5,6,11,11a‐tetrahydro‐1H‐imidazo[1′,5′:1,6]pyrido[3,4‐b]indole‐1,3(2H)‐dione as low nanomolar, orally bioavailable autotaxin inhibitor-Reference-Cited by-同舟云学术

Structure‐based discovery of ( S )‐2‐amino‐6‐(4‐fluorobenzyl)‐5,6,11,11a‐tetrahydro‐1H‐imidazo[1′,5′:1,6]pyrido[3,4‐b]indole‐1,3(2H)‐dione as low nanomolar, orally bioavailable autotaxin inhibitor

Published:2022-01-03 Issue: Volume: Page:
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Roy Ashis¹,Sarkar Tonmoy¹,Datta Sebak¹,Maiti Arup¹,Chakrabarti Monali¹,Mondal Trisha¹,Mondal Chaitali¹,Banerjee Apurba¹,Roy Subhasis¹,Mukherjee Soumen¹,Muley Pragati¹,Chakraborty Sabyasachi¹,Banerjee Manish¹,Kundu Mrinalkanti¹^ORCID,Roy Kuldeep K.²^ORCID

Affiliation:

1. TCG Lifesciences Pvt. Ltd. Kolkata India

2. Department of Pharmaceutical Sciences School of Health Sciences UPES Dehradun India

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.14017

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4. Autotaxin, a secreted lysophospholipase D, as a promising therapeutic target in chronic inflammation and cancer;Barbayianni E.;Progress in Lipid Research,2015

5. Autotaxin inhibitors: A patent review;Barbayianni E.;Expert Opinion on Therapeutic Patents,2013

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