Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin-Reference-Cited by-同舟云学术

Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin

Published:2011-06-09 Issue:13 Volume:54 Page:4619-4626
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Albers Harald M. H. G.¹,Hendrickx Loes J. D.¹,van Tol Rob J. P.¹,Hausmann Jens¹,Perrakis Anastassis¹,Ovaa Huib¹

Affiliation:

1. Division of Cell Biology, §Netherlands Proteomics Centre, and ∇Division of Biochemistry, The Netherlands Cancer Institute, Plesmanlaan 121, 1066 CX Amsterdam, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200310q

Reference24 articles.

1. Identification of Human Plasma Lysophospholipase D, a Lysophosphatidic Acid-producing Enzyme, as Autotaxin, a Multifunctional Phosphodiesterase

2. Autotaxin has lysophospholipase D activity leading to tumor cell growth and motility by lysophosphatidic acid production

3. The ins and outs of lysophosphatidic acid signaling

4. Autotaxin, an ectoenzyme that produces lysophosphatidic acid, promotes the entry of lymphocytes into secondary lymphoid organs

5. Regulation and biological activities of the autotaxin–LPA axis

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