BU08073 a buprenorphine analogue with partial agonist activity at μ-receptorsin vitrobut long-lasting opioid antagonist activityin vivoin mice
Author:
Affiliation:
1. SRI International; Menlo Park CA USA
2. Torrey Pines Institute for Molecular Studies; Port St. Lucie FL USA
3. Department of Pharmacy and Pharmacology; University of Bath; Bath UK
Funder
National Institute on Drug Abuse
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/bph.12796/fullpdf
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5. Long-acting kappa opioid antagonists disrupt receptor signaling and produce noncompetitive effects by activating c-Jun N-terminal kinase;Bruchas;J Biol Chem,2007
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